Библиотеки химических соединений для ин витро скрининга (HTS)
Научно-исследовательский институт ХимРар предлагает услуги по ин силико и ин витро высокопроизводительному скринингу (high-throughput screening, HTS) биологической активности индивидуальных соединений и библиотек разнообразных химических соединений.
В наличии коллекция в 1.6 миллиона соединений (diverse collection):
- Discovery chemistry public available >4Y old (DC) – 1,000,000
- New chemistry public available 3 Y old (NC) – 485,000 соединений
- Innovative chemistry non-exclusive 1Y old (IC ) – 120,000 соединений
Список доступных для ин витро скрининга библиотек соединений
Новые библиотеки (2020):
- 3D-Pharmacophore Based Diversity Library -52,000 соединений
- Opportunistic Pathogens of Immunocompromised Hosts Annotated Library – 2,100 соединений
- RNA-Protein Interaction Inhibitors Library – 2,111 соединений
- Cysteine Targeted Covalent Library – 41,378 соединений
- 300k Representative Соединений Library (Bemis-Murcko Algorithm) – 300,000 соединений
- Antiviral Annotated Library – 22,775 соединений
- PLpro Library – 6,442 соединений
- 3CLpro Library – 4,871 соединений
- ACE2 Library – 3,117 соединений
- MCL1 Targeted Library Selection – 12,000 соединений
- Arginase Targeted Library – 2,000 соединений
- Chelators targeting matrix metalloproteinases library – 9,300 соединений
- Ion Channels Focused Library – 26,000 соединений
- Histone Deacetylases (HDAC) Targeted Library Selection – 9,500
- CNS Annotated Library – 733 соединений
- PTPN-targeted-library Library – 33,000 соединений
- CORONAVIRUS Library – 21,145 соединений
- Lipid Metabolism Library – 9,000 соединений
- Human Phosphatases Annotated Library – 225 соединений
- Human Receptors Annotated Library – 5,600 соединений
- Purine Based Nucleoside Library – 1,300 соединений
- STING Agonist Library – 6,000 соединений
- Nucleoside Mimetics Library – 2,600 соединений
- RPTP Targeted Library – 3,900 соединений
- Human Transcription Factors Annotated Library – 5,278 соединений
- Human Proteases Annotated Library – 3,000 соединений
- Human Kinases Annotated Library – 2,500 соединений
- Human Ion Channels Annotated Library – 400 соединений
- Human GPCR Annotated Library – 5,800 соединений
- Regenerative Medicine Focused Library – 23,000 соединений
- Selective Target Activity Profiling library – 18,000 соединений
- Neurotransmitter Transporter Inhibitors library – 12,000 соединений
- MCE-18 Trends in Medicinal Chemistry – 50,000 соединений
- Epitranscriptome Focused Small Molecule Library – 21,000 соединений
- Cardiovascular Library – 23,000 соединений
- RNA Isosteric Trinucleotide Mimetics Library – 29,000 соединений
- Protein Kinases Inhibitors Library – 38,000 соединений
- Antibacterial соединений library – 15,000 соединений
- Therapeutical Diversity Annotated Library – 2,000 соединений & 6,500 соединений
- Covalent inhibitors Library – 12,000 соединений
Аннотированные библиотеки:
- Antiviral Annotated Library – 22,775 соединений
- CNS Targets Activity Set – 7,000 соединений
- Therapeutical Diversity Annotated Library – 2,000 соединений & 6,500
- 3D-Biodiversity Library – 34,000 соединений
- Target Identification, Phenotypic Screening Library (TIPS) – 35,000
- Launched & Clinically Evaluated Drugs Library – 274 соединений
- ChemoGenomic Annotated library for Phenotypic Screening – 99,000
- Selective Target Activity Profiling library – 18,000 соединений
- Human GPCR Annotated Library – 5,800 соединений
- Human Ion Channels Annotated Library – 400 соединений
- Human Kinases Annotated Library – 2,500 соединений
- Human Proteases Annotated Library – 3,000 соединений
- Human Transcription Factors Annotated Library – 5,300 соединений
- Human Receptors Annotated Library – 5,600 соединений
- Human Phosphatases Annotated Library – 225 соединений
- CNS Annotated Library – 773 соединений
- Opportunistic Pathogens of Immunocopromised Hosts Annotated Library – 2,100 соединений
Разнообразные библиотеки (Diversity libraries):
- 3D-Pharmacophore Based Diversity Library -52,000 соединений
- 3D-Diversity Natural-Product-Like Library -21,000 соединений
- Representative Diversity libraries out of 1,6M stock – 50,000 соединений, 100,000 соединений, 150,000 соединений
- 300k Representative Соединений Library (Bemis-Murcko Algorithm) – 300,000 соединений
- SmartTM Library – 54,000 соединений
- Soluble Diversity Library – 9,500 соединений
- MEC-18 Trends in Medicinal Chemistry – 50,000 соединений
- Targeted Diversity Library – 45,429 соединений
Фокусированные библиотеки:
- PPI CDI Library – 230,000 соединений
- PPI Helix Turn 3D-Mimetics Library – 74,000 соединений
- PPI Tripeptide Mimetics Library – 25,000 соединений
- Peptidomimetic Library – 38,400 соединений
- PDZ PPI Library – 4,000 соединений
- Nonpeptide Peptidomimetics PPI library – 22,000 соединений
- Eccentric PPI Library – 13,000 соединений
- Cyclic Ugi PPI Library – 10,000 соединений
- Alpha-Helix Mimetics Library– 28,000 Соединений
- Peptidomimetics of Beta-Turn Motifs Library – 2,679 соединений
- Macrocycles Library – 3,300 соединений
- 3D Mimetics PPI Library – 2,000 соединений
- Recognition Elements PPI Library – 26,000 соединений
- Bcl2-PPI Inhibitors Library – 11,000 соединений
- Library of Small Molecule Inhibitors of beta-Catenin Signaling – 8,000
- MDM2-p53 interaction inhibitors Library – 23,000 соединений
- SH2 Library – 12,000 соединений
- Library of Small Molecule Modulators & Inhibitors of Bromodomains – 5,816 соединений
- DGK Inhibitors Library – 12,000 соединений
- Focused Epigenetics Set – 30,431 соединений
- Hsp90-Targeted Library – 13,000 соединений
- SH2 PTB Focused Library – 7,000 соединений
- Nucleoside Mimetics Library – 2,600
- Purine Based Nucleoside Library – 1,300 соединений
- CNS MPO Library – 30,000 соединений
- CNS Targets Library – 44,000 соединений
- CNS targets activity set – 7,000 соединений
- CNS Library – 26,000 соединений
- CNS BBB Library – 23,000 соединений
- CNS Annotated Library – 773 соединений
- GABA library – 17,915 соединений
- Purinergic Library – 3,500 соединений
- Neurotransmitter Transporter Inhibitors library – 12,000 соединений
- Ion Channels Focused Library – 26,000 соединений
- Ligand-Gated Ion Channels Library – 4,000 соединений
- Voltage-Gated Ion Channel-Targeted Library – 5,000 соединений
- GPCR Target Platform Library – 40,000 соединений
- PTPN-targeted-library Library – 33,000 соединений
- Protein Kinases Inhibitors Library – 38,000 соединений
- Akt-Targeted Library – 12,000 соединений
- Allosteric Kinases Inhibitors Library – 26,000 соединений
- Aurora A-B Kinases Library – 10,000 соединений
- KRAS-Targeted Library – 11,000 соединений
- Proline Kinase Library – 2,000 соединений
- Type II Kinase Inhibitors Library – 8,000 соединений
- C-Met Library – 16,000 соединений
- PI3K-Targeted Library – 19,000 соединений
- Antiviral Annotated Library – 22,775 соединений
- PLpro Library – 6,442 соединений
- ACE2 Library – 222 compound
- 3CLpro Library – 4,871 соединений
- Antiviral Library – 87,043 соединений
- Anti-HIV1 Library – 21,000 соединений
- Antiviral HBV – 11,000 соединений
- CORONAVIRUS Library – 21,145 соединений
- Androgen Receptor Antagonists Library – 4,300 соединений
- RAR (Nuclear receptors) Ligands Library – 6,000 соединений
- Anticancer Library – 65,000 соединений
- Antimitotic Tubulin Library – 18,000 соединений
- Histone Deacetylases (HDAC) Targeted Library Selection – 9,500
- Developmental Pathway (Hh/Wnt) Set – 2,000 соединений
- MEF2-HDAC (class II) Modulators Library – 6,000 соединений
- Arginase Targeted Library – 2,000 соединений
- Chelators targeting matrix metalloproteinases library – 9,300 соединений
- MCL1 Targeted Library Selection – 12,000 соединений
- Cysteine Proteases Inhibitors Library – 8,000 соединений
- Serine Proteases Inhibitors Library – 37,000 соединений
- PRMT Library – 31,000 соединений
- Immunological Library – 7,300 соединений
- PD-1/L1 Library – 500 соединений
- TLR-8 ligands Library – 900 соединений
- Anti-Inflammatory Library – 28,000 соединений
- Cardiovascular Library – 23,000 соединений
- Lipid Metabolism Library – 9,000 соединений
- Anti-Aging Library – 50,000 Соединений
- Regenerative Medicine Focused Library – 23,000 соединений
- Autophagy-Targeted Library – 17,000 соединений
- RNA Isosteric Trinucleotide Mimetics Library – 29,000 соединений
- Chemokines Library – 20,000 соединений
- Angiogenesis library – 17,000 соединений
- BRD4 targeted library – 5,000 соединений
- Integrin Receptors Targeted library – 2,000 соединений
- Indoleamine 2,3-dioxygenase 1 focused library – 6,000 соединений
- Neuropeptide S Library – 3,000 соединений
- RNA-Protein Interaction Inhibitors Library – 2,111 соединений
- Nucleic acid ligands – 9,000 соединений
- RAR (Nuclear receptors) Ligands Library – 6,000 соединений
- Epitranscriptome Focused Small Molecule Library – 21,000 соединений
- RPTP Targeted Library – 3,900 соединений
- Adenosine Receptors Targeted Library – 21,000 соединений
- Glucocorticoid receptors Library – 5,000 соединений
- Macl-GPIb alpha Interaction Library – 27,000 соединений
- STING Agonist Library – 6,000
- Antiparasite library – 28,000 соединений
- Anti-infective Library – 20,600 соединений
- Antibacterial соединений library – 15,000 соединений
- Covalent inhibitors Library – 12,000 соединений
- Cysteine Targeted Covalent Library – 41,378 соединений
- New Agro Library – 50,000 соединений
- Antifungal Library – 18,000 соединений
- Beyond the Flatland Library sp3 enriched – 100,000 соединений
- Spiro-library – 19,000 соединений
- Indole Derivatives – 12,000 соединений
- 3D-Diversity Natural-Product-Like Library – 21,000 соединений
- Natural-Product-Based Library – 4,000 соединений
- Natural Соединений Library – 374 соединений
- Steroid-like-соединений – 543 соединений
- 3D-Fragment-Library – 4,500 соединений
- Fragments Library – 13,000 соединений
- Dark Chemical Matter Library – 25,000 Соединений
- Frequent Hitters Library – 9,000 соединений
Список библиотек регулярно обновляется.
Для получения актуальной информации по наличию и условиях продажи библиотек и/или услуг по ин силико и ин витро скринингу вы можете отправить запрос на email указанный ниже.